Synthesis and Diels–Alder Reactivity of 4-Fluoro-4-Methyl-4H-Pyrazoles
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چکیده
منابع مشابه
4-(4-Methoxyphenyl)-4-methyl-2,6-diphenyl-4H-thiopyran
The asymmetric unit of the title compound, C(25)H(22)OS, comprises two similar 4-(4-methoxy-phen-yl)-4-methyl-2,6-diphenyl-4H-thio-pyran mol-ecules. In each, the six-membered thio-pyran ring adopts a planar conformation (r.m.s. deviation of 0.041Å for the ring in one mol-ecule and 0.008 Å in the other). The methoxy-phenyl substituent is in a pseudo-axial position. The crystal studied is an inve...
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A series of 3-alkoxy-4-(4-(hexyloxy/heptyloxy) phenyl)-4H-1,2,4-triazole was synthesized. The anticonvulsant effect and neurotoxicity of the compounds were calculated with maximal electroshock (MES) test and rotarod tests with intraperitoneally injected mice. Among the synthesized compounds, compound 3-heptyloxy-4-(4-(hexyloxy) phenyl)-4H-1,2,4-triazole (5f) was the most active one and also had...
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ژورنال
عنوان ژورنال: International Journal of Molecular Sciences
سال: 2020
ISSN: 1422-0067
DOI: 10.3390/ijms21113964